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levenabiopharma產(chǎn)品目錄

更新時(shí)間:2021-01-08      點(diǎn)擊次數(shù):2083

 

 levenabiopharma用于連接抗體和藥物的連接子

levenabiopharma生物制藥提供不同結(jié)構(gòu)和功能的多種連接子,可用于抗體和藥物的偶聯(lián)的連接子。更重要的是,聯(lián)寧自主開(kāi)發(fā)的擁有*知識(shí)產(chǎn)權(quán)的連接子可以將藥物可控地偶聯(lián)到抗體上,更易實(shí)現(xiàn)批次間的產(chǎn)品質(zhì)量控制。為更好地支持客戶的藥物開(kāi)發(fā),levenabiopharma還提供連接子定制設(shè)計(jì)和合成服務(wù)。

levenabiopharma產(chǎn)品目錄

 

產(chǎn)品目錄號(hào)產(chǎn)品名稱Cas 號(hào)純度可提供數(shù)量
VC1001Val-Cit-PAB159857-79-195%mg - 500g
VC1002Fmoc-Val-Cit-PAB159858-22-795%mg - 500g
VC1003Fmoc-Val-Cit-PAB-PNP863971-53-395%mg - 500g
VC1004MC-Val-Cit-PAB-PNP159857-81-595%mg-100g
FK1001Phe-Lys(Trt)-PAB 95%mg - kg
FK1002Fmoc-Phe-Lys(Trt)-PAB 95%mg - kg
FK1003Fmoc-Phe
-Lys(Trt)-PAB-PNP
1116086-09-995%mg - kg
AN1001Ala-Ala-Asn-PAB TFA salt 95%mg - kg
AN1002Fmoc-Ala-Ala-Asn-PAB-PNP 95%mg - kg
H1001Fmoc-Gly3-Val-Cit-PAB 95%mg-100g
H1002Fmoc-Gly3-Val-Cit-PAB-PNP 95%mg-100g
D1000SMCC64987-85-598%500mg-500g
DS1001Py-ds-Prp-OSu 95%mg - kg
DS1003Py-ds-dmBut-OSu 95%mg - 100g
DS1013Py-ds-dmBut-OPFP 95%mg - 100g
DS1011Py-ds-Prp-OPFP 95%mg - kg
MA1000MAL-HA-OSu 95%mg - kg
MA2011MAL-di-EG-OPFP 95%mg - kg
MA2012MAL-tri-EG-OPFP 95%mg - kg
MA2013MAL-tetra-EG-OPFP 95%mg - kg
AZ1011N3-di-EG-OPFP 95%mg - kg
AZ1012N3-tri-EG-OPFP 95%mg - kg
AZ1013N3-tetra-EG-OPFP 95%mg - kg
AL1001ALD-BZ-OSu 95%mg - kg
AL1003ALD-di-EG-OSu 95%mg - kg
AL1005ALD-tetra-EG-OSu 95%mg - kg
AL1013ALD-di-EG-OPFP 95%mg - kg
AL1015ALD-tetra-EG-OPFP 95%mg - kg
HA1011PHA-di-EG-OPFP 95%mg - kg
HA1013PHA-tetra-EG-OPFP 95%mg - kg

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ADC細(xì)胞毒素藥物

 

從抗體到靶向抗體藥物偶聯(lián)物的合成過(guò)程有挑戰(zhàn)性。為了設(shè)計(jì)出高效的抗體藥物偶聯(lián)物,毒素的選擇是至關(guān)重要的。聯(lián)寧生物制藥提供各種各樣的微管蛋白抑制劑和DNA烷基化試劑,這些試劑已被證實(shí)是抗體藥物偶聯(lián)物負(fù)載的有效細(xì)胞毒素。對(duì)下面列出的這些毒素, 聯(lián)寧可以提供毫克級(jí)至100克級(jí)的高質(zhì)量產(chǎn)品。

For structures, click here>>>

產(chǎn)品目錄號(hào)產(chǎn)品名稱Cas 號(hào)純度可提供數(shù)量
T1001Dolastatin 10110417-88-498%mg - 100g
T1002Monomethyl Dolastatin 10203849-91-698%mg - 100g
T1003Auristatin E160800-57-798%mg - 100g
T1004Monomethyl Auristatin E474645-27-798%mg - 100g
T1005Auristatin F163768-50-198%mg - 100g
T1006Monomethyl Auristatin F745017-94-198%mg - 100g
T1007HTI-286228266-40-895%mg - g
T1008Tubulysin M205304-86-595%mg - g
T1009Maytansinoid AP-366547-09-985%mg
T1109Maytansinol57103-68-195%mg - 100g
LN-T-4582DM1139504-50-098%mg - 100g
LN-T-7544DM4799840-96-398%mg - 10g
T1102Boc-Val-Dil-Dap-OH 95%mg - kg
T1202Boc-Val-Dil-Dap-Phe-OMe 95%mg - kg
T1222Boc-Val-Dil-Dap-Doe 95%mg - kg
T1224Boc-Val-Dil-Dap-Nrp 95%mg - kg
T1302Boc-N-Me-Val-Val-Dil-Dap-OH 95%mg - kg
T1108Tubulysin IM-1 95%mg - 100g
T1208Tubulysin IM-2 95%mg - 100g
T1308Tubulysin IM-3 95%mg - 100g
D1001Duocarmycin SA152785-82-595%mg - g
D1007Duocarmycin TM 95%mg - g
D1008Duocarmycin MA 95%mg - g
D1009Duocarmycin DM 95%mg - g
D4000Nemorubicin108852-90-095%mg - 10 g
D4001PNU-159682202350-68-3>90%mg -10 g
LN-T-6888Calicheamicin g1108212-75-5>95%mg-100mg
D4006N-Acetyl-Calicheamicin g1108212-76-6
>95%
mg-100g
D4007a-Amanitin23109-05-9>95%mg-g
D4008PBD-dimer1222490-34-7>90%mg-100mg

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易用的細(xì)胞毒素 (SET™)

聯(lián)寧生物制藥提供安全易用的毒素(SET™),這是一種可以快速篩選抗體藥物偶聯(lián)物的新型研究工具。SET™產(chǎn)品線包括很多已驗(yàn)證的連接子-毒素,分別裝入預(yù)包裝好的小瓶中。每個(gè)SET™小瓶含有約200納摩的連接子-毒素,按藥物/抗體比(DAR)為3-4計(jì)算的話, 足夠偶聯(lián)5毫克抗體。客戶不需要稱重或分裝連接子-毒素,只需按照產(chǎn)品說(shuō)明書上提供的溶解方案,即可使用SET™。SET™不僅易于使用,更重要的是可以大限度地減少實(shí)驗(yàn)過(guò)程中暴露毒素的風(fēng)險(xiǎn)。目前,SET™可用于以下類別的偶聯(lián)反應(yīng):

 

    ?胺反應(yīng)SET™ 
    ?硫醇反應(yīng)SET™ 
    ?點(diǎn)擊反應(yīng)SET™ 
    ?轉(zhuǎn)肽酶反應(yīng) SET™ 

For structures, click here>>>

胺反應(yīng) SET™  
產(chǎn)品目錄號(hào)產(chǎn)品名稱數(shù)量單價(jià)
SET0100OSu-Glu-vc-PAB-MMAE200 nmol$500
SET0101SMCC-DM1200 nmol$500
SET0102SPDB-DM4200 nmol$650
SET0103OSu-PEG4-vc-PAB-DMEA
Duocarmycin SA
200 nmol$750
SET0104Mylotarg-linker200 nmol$950
SET0105OSu-Glu-vc-PAB-MMAD200 nmol$500
SET0106Sulfo-SPDB-DM4200 nmol$950.00
SET0107IMGN779-linker200 nmol$2,200.00
SET0108OSu-PEG4-vc-PAB-DMEA
Duocarmycin TM
200 nmol$750.00
SET0109OSu-PEG4-vc-PAB-DMEA
Duocarmycin DM
200 nmol$750.00
硫醇反應(yīng)SET™  
產(chǎn)品目錄號(hào)產(chǎn)品名稱數(shù)量單價(jià)
SET0201MC-vc-PAB-MMAE200 nmol$ 500
SET0202MC-MMAF200 nmol$ 500
SET0203MC-DM1200 nmol$ 700
SET0204MC-MMD-10200 nmol$ 600
SET0205MA-PEG4-vc-PAB-DMEA-
duocarmycin SA
200 nmol$ 750
SET0206MC-vc-PAB-C6-a-amanitin200 nmol$ 850
SET0207MC-cleavable-linker-a-amanitin200 nmol$ 600
SET0208MC-vc-PAB-DMEA-(PEG2)-
duocarmycin SA
200 nmol$ 800
SET0209MC-vc-PAB-Tubulysin M200 nmol$ 800
SET0210MC-va-PAB-MMAD200 nmol$ 500
SET0211MA-PEG4-VC-PAB-DMAE-PNU159682200 nmol$ 950
SET0212MA-PEG4-VA-PBD200 nmol$ 1,100
SET0213MC-vc-PAB-MMAF200 nmol$ 500
SET0214MC-vc-PAB-MMAD200 nmol$ 500
SET0215MC-vc-PAB-Auristatin 0101200 nmol$ 900
SET0216MA-PEG8-VA-PAB-SG3199200 nmol$ 1,950
SET0217CL2A-SN 38200 nmol$ 800
SET0218MC-GGFG-DX8951200 nmol$ 950
SET0219MEDI4276_linker payload200 nmol$ 1,100
SET0220MA-PEG4-vc-PAB-DMEA-
duocarmycin TM
200 nmol$ 750
SET0221MC-vc-PAB-(PEG2)-
duocarmycin TM
200 nmol$ 900
SET0222MA-PEG4-vc-PAB-DMEA-
duocarmycin DM
200 nmol$ 750
SET0223MC-vc-PAB-(PEG2)-
duocarmycin DM
200 nmol$ 900
SET0224DGN549200 nmol$ 1,900
SET0225MPB-vc-PAB-MMAE200 nmol$ 550
SET0226MPB-MMAF200 nmol$ 550
點(diǎn)擊反應(yīng)SET™  
產(chǎn)品目錄號(hào)產(chǎn)品名稱數(shù)量單價(jià)
SET0301DBCO-PEG4-vc-PAB-MMAE200 nmol$ 650
SET0302DBCO-PEG4-MMAF200 nmol$ 750
SET0303DBCO-PEG4-Ahx-DM1200 nmol$ 750
SET0304DBCO-PEG4-vc-PAB-
Duocarmycin SA
200 nmol$ 900
SET0305DBCO-PEG4-vc-PAB-(PEG2)-
Duocarmycin SA
200 nmol$ 1,050
SET0306DBCO-PEG4-VA-PBD200 nmol$ 1,100
SET0307DBCO-PEG4-vc-PAB-MMAF200 nmol$ 650
SET0308DBCO-PEG4-vc-PAB-MMAD200 nmol$ 650
SET0309DBCO-PEG4-vc-PAB-
Duocarmycin TM
200 nmol$ 900
SET0310DBCO-PEG4-vc-PAB-(PEG2)-
Duocarmycin TM
200 nmol$ 1,050
SET0311DBCO-PEG4-vc-PAB-
Duocarmycin DM
200 nmol$ 900
SET0312DBCO-PEG4-vc-PAB-(PEG2)-
Duocarmycin DM
200 nmol$ 1,050
SET0313DBCO-PEG4-VC-PAB-DMAE-PNU159682200 nmol$ 1,050
SET0314DBCO-PEG4-DMAE-PNU159682200 nmol$ 1,000
SET0315DBCO-PEG4-GGFG-DX8951200 nmol$ 1,050
SET0316DBCO-PEG4-vc-PAB-Ahx-DM1200 nmol$ 850
SET0317DBCO-PEG8-VA-PAB-SG3199200 nmol$ 2,050
轉(zhuǎn)肽酶反應(yīng) SET™  
產(chǎn)品目錄號(hào)產(chǎn)品名稱數(shù)量單價(jià)
SET0401Gly3-vc-PAB-MMAE200 nmol$850
SET0402Gly3-MMAF200 nmol$850
SET0403Gly5-Ahx-DM1200 nmol$950
SET0404PNU159682-EDA-Gly3200 nmol$1,100

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ADC篩選試劑盒

 

 

聯(lián)寧生物制藥提供研究階段抗體藥物偶聯(lián)物體外活性的篩選服務(wù)。公司的細(xì)胞庫(kù)擁有超過(guò)100個(gè)癌細(xì)胞株,可以幫助客戶評(píng)估抗體藥物偶聯(lián)物的細(xì)胞毒性和治療潛力。公司還可以根據(jù)客戶的需求靈活安排用這些細(xì)胞株來(lái)篩選抗體藥物偶聯(lián)物。

 

聯(lián)寧生物制藥制備了目前市面上常用的抗體藥物偶聯(lián)物,如T-DM1,brentuximab vedotin,VEGR2-ADC等,作為抗體藥物偶聯(lián)物評(píng)估的對(duì)照物,為客戶評(píng)估抗體藥物偶聯(lián)物生物仿制藥提供方便。

聯(lián)寧生物制藥開(kāi)發(fā)的以蛋白A和蛋白G的PSKA™和PSKG™的抗體藥物偶聯(lián)物預(yù)篩選試劑盒,在不做偶聯(lián)的情況下, 可以快速鑒定適合抗體藥物偶聯(lián)物研發(fā)用的抗體。使用這些試劑盒,可以直接篩選初級(jí)抗體,略去單獨(dú)將毒素偶聯(lián)到抗體上的過(guò)程。我們提供的PSK篩選試劑盒包括業(yè)界常用毒素,如MMAE,MMAF,DM1和duocarmycin。

產(chǎn)品目錄號(hào)產(chǎn)品名稱產(chǎn)品說(shuō)明數(shù)量單價(jià)
LEV-PSKA-100ADC pre-screening kit AFour vials containing Protein A preloaded with
1x MMAE (cleavable linker) 
1x MMAF (non-cleavable linker) 
1x MCC-DM1 (non-cleavable linker)
1x Duocarmycin (cleavable linker)
4x100 µL$ 900.00
LEV-ADM-100Protein A-DM1Protein A preloaded with MCC-DM1 (non-cleavable linker)100 µL$ 300.00
LEV-AME-100Protein A-MMAEProtein A preloaded with MMAE (cleavable linker)100 µL$ 300.00
LEV-AMF-100Protein A-MMAFProtein A preloaded with MMAF (non-cleavable linker)100 µL$ 300.00
LEV-ADC-100Protein A-DuocarmycinProtein A preloaded with Duocarmycin (cleavable linker)100 µL$ 400.00
LEV-ACC-100Protein A-CalicheamicinProtein A preloaded with Calicheamicin (cleavable linker)100 µL$ 400.00
LEV-APB-100Protein A-PBDProtein A preloaded with PBD100 µL$ 400.00
LEV-PSKG-100ADC pre-screening kit GFour vials containing Protein A preloaded with
1x MMAE (cleavable linker) 
1x MMAF (non-cleavable linker) 
1x MCC-DM1 (non-cleavable linker)
1x Duocarmycin (cleavable linker)
4x100 µL$ 900.00
LEV-GDM-100Protein G-DM1Protein G preloaded with MCC-DM1 (non-cleavable linker)100 µL$ 300.00
LEV-GME-100Protein G-MMAEProtein G preloaded with MMAE (cleavable linker)100 µL$ 300.00
LEV-GMF-100Protein G-MMAFProtein G preloaded with MMAF (non-cleavable linker)100 µL$ 300.00
LEV-GDC-100Protein G-DuocarmycinProtein G preloaded with Duocarmycin (cleavable linker)100 µL$ 400.00
LEV-GAM-100Protein G-AmanitinProtein G preloaded with Amanitin (cleavable linker)100 µL$ 400.00
LEV-GAL-100Protein G-AmanitinProtein G preloaded with Amanitin (Levena cleaveable linker)100 µL$ 400.00

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抗細(xì)胞毒性藥物抗體

 

 

聯(lián)寧生物制藥開(kāi)發(fā)了各種抗細(xì)胞毒性藥物抗體用來(lái)支持客戶的臨床前藥物研究。目前,提供的抗體包括針對(duì)不同類別的細(xì)胞毒性藥物的抗毒素(藥物)單克隆和多克隆抗體。這些產(chǎn)品僅限于科研,不能用于臨床診斷

產(chǎn)品目錄號(hào)產(chǎn)品名稱毒素類型微升單價(jià)毫克/毫升
LEV-PAE1-100Rabbit Anti-vc-PAB-MMAE pAbTubulin Inhibitor100 $    500.001
LEV-PAE1-500500 $ 1,875.00
LEV-MAE1-100Mouse Anti-vc-PAB-MMAE mAb (B11F11)Tubulin Inhibitor100 $    900.001
LEV-MAE1-500500 $ 3,375.00
LEV-PAF1-100Rabbit Anti-MMAF pAbTubulin Inhibitor100 $    500.001
LEV-PAF1-500500 $ 1,875.00
LEV-MAF1-100Mouse Anti-MMAF mAb (F3B11)Tubulin Inhibitor100 $    900.001
LEV-MAF1-500500 $ 3,375.00
LEV-MAE3-100Mouse Anti-MMAE / F mAb (B12A2)Tubulin Inhibitor100 $    900.001
LEV-MAE3-500500 $ 3,375.00
LEV-MAF3-100Mouse Anti-MMAE /F mAb (C12A1)Tubulin Inhibitor100 $    900.001
LEV-MAF3-500500 $ 3,375.00
LEV-PDM1-100Rabbit Anti-DM1/4 pAbTubulin Inhibitor100 $    500.001
LEV-PDM1-500500 $ 1,875.00
LEV-MDM1-100Mouse Anti-DM1/4 mAb (F1D5)Tubulin Inhibitor100 $    900.001
LEV-MDM1-500500 $ 3,375.00
LEV-MDM2-100Mouse Anti-DM1/4 mAb (G2F3)Tubulin Inhibitor100 $    900.001
LEV-MDM2-500500 $ 3,375.00
LEV-PCA1-100Rabbit Anti-Calicheamicin pAbDNA Damaging100 $    750.000.5
LEV-PCA1-500500 $ 2,800.00
LEV-MCA1-100Mouse Anti-Calicheamicin mAb (B1G9)DNA Damaging100 $ 1,250.000.5
LEV-MCA1-500500 $ 4,700.00
LEV-MCA2-100Mouse Anti-Calicheamicin mAb (C1F12) DNA Damaging100 $ 1,250.000.5
LEV-MCA2-500500 $ 4,700.00
LEV-PDU1-100Rabbit Anti-Duocarmycin pAb DNA Damaging100 $    750.000.5
LEV-PDU1-500500 $ 2,800.00
LEV-MDU3-100Mouse Anti-Duocarmycin mAb (E11A1) DNA Damaging100 $    900.000.5
LEV-MDU3-500500 $ 3,375.00
LEV-MDU1-100Mouse Anti-Duocarmycin mAb (H7A9)DNA Damaging100 $    900.000.5
LEV-MDU1-500500 $ 3,375.00
LEV-MDU2-100Mouse Anti-Duocarmycin mAb (E6B3) DNA Damaging100 $    900.000.5
LEV-MDU2-500500 $ 3,375.00
LEV-PPN1-100Rabbit Anti-PNU-159682 pAbDNA Damaging100 $    750.000.5
LEV-PPN1-500500 $ 2,800.00
LEV-MPN1-100Mouse Anti-PNU-159682 mAb (F7F2)DNA Damaging100 $    900.000.5
LEV-MPN1-500500 $ 3,375.00
LEV-MPN2-100Mouse Anti-PNU-159682 mAb (C1E3)DNA Damaging100 $    900.000.5
LEV-MPN2-500500 $ 3,375.00
LEV-MPN3-100Mouse Anti-PNU-159682 mAb (D12H11)DNA Damaging100 $    900.000.5
LEV-MPN3-500500 $ 3,375.00
LEV-PAM1-100Rabbit Anti-Amanitin pAbRNA Polymerase II and III Inhibitor100 $    650.000.5
LEV-PAM1-500500 $ 2,450.00
LEV-MAM1-100Mouse Anti-Amanitin mAb (H3E1)RNA Polymerase II and III Inhibitor100 $ 1,100.000.5
LEV-MAM1-500500 $ 4,100.00
LEV-MAM2-100Mouse Anti-Amanitin mAb (H12D6)RNA Polymerase II and III Inhibitor100 $ 1,100.000.5
LEV-MAM2-500500 $ 4,100.00
LEV-MAM3-100Mouse Anti-Amanitin mAb (C2C4)RNA Polymerase II and III Inhibitor100 $ 1,100.000.5
LEV-MAM3-500500 $ 4,100.00
LEV-PSN1-100Rabbit Anti-SN38 pAbDNA Topoisomerase I Inhibitor100 $    650.000.5
LEV-PSN1-500500 $ 2,450.00
LEV-MSN1-100Mouse Anti-SN38 mAb (10F11A9D6)DNA Topoisomerase I Inhibitor100 $    900.000.5
LEV-MSN1-500500 $ 3,375.00
LEV-MSN2-100Mouse Anti-SN38 mAb (8E10F12F3)DNA Topoisomerase I Inhibitor100 $    900.000.5
LEV-MSN2-500500 $ 3,375.00
LEV-MSN3-100Mouse Anti-SN38 mAb (8E10A4A1)DNA Topoisomerase I Inhibitor100 $    900.000.5
LEV-MSN3-500500 $ 3,375.00
LEV-PSG1-100Rabbit Anti-PBD SG3199 pAb DNA Inhibitor                                100 $    900.000.5
LEV-PSG1-500500 $ 3,374.00
LEV-MSG1-100Mouse Anti-PBD SG3199 (7H6H9A6) mAbDNA Inhibitor100 $ 1,250.000.5
LEV-MSG1-500500 $ 4,500.00
LEV-MSG2-100Mouse Anti-PBD SG3199 (8G2H12A9) mAbDNA Inhibitor100 $ 1,250.000.5
LEV-MSG2-500500 $ 4,500.00
LEV-MSG3-100Mouse Anti-PBD SG3199 (8B3D12G1) mAbDNA Inhibitor100 $ 1,250.000.5
LEV-MSG3-500500 $ 4,500.00

 

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